Skip to main content
Skip to main content

The Synthesis and Dynamic Covalent Chemistry of Amidoboronates

 

BN containing heterocycles can give access to different and interesting reactivity as well as functionality compared to their carbon analogues. Amidoboronates are a novel class of BN containing heterocycles readily synthesised from N-aryl iminoboronates through a reductive coupling using a single electron reductant (Dalton Trans., 2023 , 52, 9189 - 9201). 
The reductive coupling yields up to 3 different amidoboronate isomers, the diastereomeric rac5 and meso5 products and the fused six-membered rac6 ring system (Chem. Eur. J., 2018 , 24 , 1200 - 12005). Amidoboronates potentially contain up to 3 types of dynamic covalent bonds including previously unknown dynamic B-N bonds. We have shown that the rac5/rac6 isomeric ratio can be influenced through variation of the para-aniline substituent and catechol sub-components through exploitation of the dynamic covalent B-N and B-O bonds (ChemPlusChem, 2022 , 87 , e20220022).  

Amidoboronates
Amidoboronates2

Figure from ChemPlusChem, 2022 , 87, e20220022